Ulcerative colitis

Active Ingredient: Guselkumab

Indication for Guselkumab

Population group: only adults (18 years old or older)
Therapeutic intent: Curative procedure

Guselkumab is indicated for the treatment of adult patients with moderately to severely active ulcerative colitis who have had an inadequate response, lost response, or were intolerant to either conventional therapy, or a biologic treatment.

For this indication, competent medicine agencies globally authorize below treatments:

200 mg administered intravenously at Week 0, 4 and 8, and thereafter 100 mg administered subcutaneously at Week 16 and every 8 weeks or 200 mg at Week 12 and every 4 weeks

For:

Dosage regimens

Regimen A: Intravenous, 200 milligrams guselkumab, once every 4 weeks, 3 doses in total, over the duration of 16 weeks. Afterwards, subcutaneous, 100 milligrams guselkumab, once every 8 weeks.

Regimen B: Intravenous, 200 milligrams guselkumab, once every 4 weeks, 3 doses in total, over the duration of 16 weeks. Afterwards, subcutaneous, 200 milligrams guselkumab, once every 4 weeks.

Detailed description

The recommended induction dose is 200 mg administered by intravenous infusion at Week 0, Week 4 and Week 8.

After completion of the induction dose regimen, the recommended maintenance dose starting at Week 16 is 100 mg administered by subcutaneous injection every 8 weeks (q8w). Alternatively, for patients who do not show adequate therapeutic benefit to induction treatment according to clinical judgement, a maintenance dose of 200 mg administered by subcutaneous injection starting at Week 12 and every 4 weeks (q4w) thereafter, may be considered.

Immunomodulators and/or corticosteroids may be continued during treatment with guselkumab. In patients who have responded to treatment with guselkumab, corticosteroids may be reduced or discontinued in accordance with standard of care.

Consideration should be given to discontinuing treatment in patients who have shown no evidence of therapeutic benefit after 24 weeks of treatment.

Missed dose

If a dose is missed, the dose should be administered as soon as possible. Thereafter, dosing should be resumed at the regular scheduled time.

Elderly

No dose adjustment is required.

There is limited information in patients aged ≥65 years and very limited information in patients aged ≥75 years.

Dosage considerations

Sites for subcutaneous injection include the abdomen, thigh and back of the upper arm. Guselkumab should not be injected into areas where the skin is tender, bruised, red, hard, thick or scaly. If possible, areas of the skin that show psoriasis should be avoided as injection sites.

Active ingredient

Guselkumab

Guselkumab is a human IgG1λ monoclonal antibody (mAb) that binds selectively to the interleukin 23 (IL-23) protein with high specificity and affinity. IL-23 is a cytokine that is involved in inflammatory and immune responses. By blocking IL-23 from binding to its receptor, guselkumab inhibits IL-23-dependent cell signalling and release of proinflammatory cytokines.

Read more about Guselkumab

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