Insect stings, insect bites, nettle stings

Active Ingredient: Mepyramine

Indication for Mepyramine

Population group: only children (1 year - 12 years old) , adolescents (12 years - 18 years old) , adults (18 years old or older)

Symptomatic relief of skin irritation caused by insect stings, insect bites and nettle stings.

For this indication, competent medicine agencies globally authorize below treatments:

3 spreads in 3 divided doses daily

Route of admnistration

Cutaneous

Defined daily dose

3 - 3 {spreads}

Dosage regimen

From 1 To 1 {spreads} 3 time(s) per day every day

Active ingredient

Mepyramine

Mepyramine is a first generation antihistamine, targeting the H1 receptor. However, it rapidly permeates the brain and so often causes drowsiness as a side effect. Mepyramine is a histamine H1 receptor inverse agonist. It binds to a G protein-coupled form of the receptor and promotes a G protein-coupled inactive state of the H1 receptor that interferes with the Gq/11-mediated signaling. Mepyramine competes with histamine for binding at H1-receptor sites on the effector cell surface, resulting in suppression of histaminic edema, flare, and pruritus. The sedative properties of mepyramine occur at the subcortical level of the CNS. It has mild hypnotic properties and some local anesthetic action and is used for allergies (including skin eruptions) both parenterally and locally. It is a common ingredient of cold remedies.

Read more about Mepyramine

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