PRODUODOPA Solution for infusion Ref.[116798] Active ingredients: Carbidopa Levodopa Levodopa and Carbidopa

Source: Health Products Regulatory Authority (IE)  Revision Year: 2024  Publisher: AbbVie Limited, Citywest Business Campus, Dublin 24, Ireland

Product name and form

Produodopa 240 mg/ml + 12 mg/ml solution for infusion.

Pharmaceutical Form

Solution for infusion (infusion).

Produodopa is a clear to slightly opalescent solution in a glass vial. The solution should be free from particulates. Produodopa may vary from colourless to yellow to brown and may have a purple or red tint. Variations in colour are expected and have no impact on product quality. The solution may become darker in colour after piercing of the vial stopper or while in the syringe.

The pH is approximately 7.4. Osmolality is approximately 2200 to 2500 mOsmol/kg but may range up to 2700 mOsmol/kg.

Qualitative and quantitative composition

1 ml contains 240 mg foslevodopa and 12 mg foscarbidopa.

10 ml contain 2400 mg foslevodopa and 120 mg foscarbidopa.

Foslevodopa and foscarbidopa are prodrugs equivalent to approximately 170 mg levodopa and 9 mg carbidopa per 1 ml.

Excipient with known effect:

Produodopa contains approximately 1.84 mmol (42.4 mg) sodium per ml.

For the full list of excipients, see section 6.1.

Active Ingredient

Carbidopa is a peripheral aromatic amino acid decarboxylase inhibitor. It prevents metabolism of levodopa to dopamine in the peripheral circulation, ensuring that a higher proportion of the dose reaches the brain, where dopamine exerts its therapeutic effects. A lower dose of levodopa can be used when it is coadministered with carbidopa, reducing the incidence and severity of peripheral side effects.

Levodopa is a precursor of dopamine, and is given as dopamine replacement therapy in Parkinson's disease.

Levodopa is a precursor of dopamine, and is given as replacement therapy in Parkinson's disease. Carbidopa is a peripheral dopa decarboxylase inhibitor. It prevents metabolism of levodopa to dopamine in the peripheral circulation, ensuring that a higher proportion of the dose reaches the brain, where dopamine acts. A lower dose of levodopa can be used, reducing the incidence and severity of side-effects.

List of Excipients

Sodium hydroxide 10N (for pH adjustment)
Hydrochloric acid, concentrated (for pH adjustment)
Water for injections

Pack sizes and marketing

Total amount of 10 ml in type I clear, colourless glass vial fitted with a grey rubber stopper, aluminium crimp cap, and turquoise plastic flip-off cap, carton with 7 vials.

Sterile, single-use infusion components (syringe, infusion set, and vial adapter) qualified for use are provided separately.

The Vyafuser pump is provided separately.

Marketing authorization holder

AbbVie Limited, Citywest Business Campus, Dublin 24, Ireland

Marketing authorization dates and numbers

PA1824/002/003

Date of first authorisation: 23rd September 2022

Drugs

Drug Countries
PRODUODOPA Austria, Cyprus, Estonia, Croatia, Israel, Romania

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