Avapritinib

Chemical formula: C₂₆H₂₇FN₁₀  Molecular mass: 498.57 g/mol  PubChem compound: 118023034

Therapeutic indications

Avapritinib is indicated for:

Unresectable or metastatic gastrointestinal stromal tumour (GIST)

Population group: only adults (18 years old or older)

Avapritinib is indicated as monotherapy for the treatment of adult patients with unresectable or metastatic gastrointestinal stromal tumours (GIST) harbouring the platelet-derived growth factor receptor alpha (PDGFRA) D842V mutation.

For this indication, competent medicine agencies globally authorize below treatments (click for details):

Advanced systemic mastocytosis (AdvSM)

Population group: only adults (18 years old or older)

Avapritinib is indicated as monotherapy for the treatment of adult patients with aggressive systemic mastocytosis (ASM), systemic mastocytosis with an associated haematological neoplasm (SM-AHN) or mast cell leukaemia (MCL), after at least one systemic therapy.

For this indication, competent medicine agencies globally authorize below treatments (click for details):

Indolent systemic mastocytosis (ISM)

Population group: only adults (18 years old or older)

Avapritinib is indicated for the treatment of adult patients with indolent systemic mastocytosis (ISM) with moderate to severe symptoms inadequately controlled on symptomatic treatment.

For this indication, competent medicine agencies globally authorize below treatments (click for details):

Contraindications

Avapritinib is contraindicated in the following cases:

Lactation

Lactation

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Factors such as age, gender, and health history are evaluated to create a personalized medication regimen.

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