Azelastine
Chemical formula: C₂₂H₂₄ClN₃O Molecular mass: 381.898 g/mol PubChem compound: 2267
Active ingredient description
Azelastine, a phthalazinone derivative is classified as a potent long-acting anti-allergic compound with selective H1 antagonist properties. An additional anti-inflammatory effect could be detected after topical ocular administration. Data from in vivo (pre-clinical) and in vitro studies show that azelastine inhibits the synthesis or release of the chemical mediators known to be involved in early and late stage allergic reactions e.g. leukotriene, histamine, PAF and serotonin.
Medicine classification
This medicinal substance has been classified in the anatomical therapeutic chemical (ATC) classification according to its main therapeutic use as follows:
Product monographs
Competent medicine agencies globally have authorized commercialization of this active ingredient according to these medication package inserts (MPIs):
Medicines
Azelastine is an active ingredient of these brands:
United States (US)
Austria (AT)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- ALLERGODROP as AZELASTINE HYDROCHLORIDE
- ALLERGOSPRAY as AZELASTINE HYDROCHLORIDE
- ASTEPRO as AZELASTINE HYDROCHLORIDE
- AZEDIL as AZELASTINE HYDROCHLORIDE
- AZELA-VISION as AZELASTINE HYDROCHLORIDE
- VIVIDRIN AZELASTIN as AZELASTINE HYDROCHLORIDE
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
- (combination) SYNAZE as AZELASTINE HYDROCHLORIDE
Brazil (BR)
- AZNITE as AZELASTINE HYDROCHLORIDE
- RINO-LASTIN as AZELASTINE HYDROCHLORIDE
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
Canada (CA)
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
Ecuador (EC)
Estonia (EE)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- (combination) BILENI as AZELASTINE HYDROCHLORIDE
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
- (combination) DYVISTANIL as AZELASTINE HYDROCHLORIDE
- (combination) SYCARA
Finland (FI)
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
France (FR)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
- (combination) SYNAZE as AZELASTINE HYDROCHLORIDE
Hong Kong (HK)
Ireland (IE)
Lithuania (LT)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- (combination) BILENI as AZELASTINE HYDROCHLORIDE
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
Malta (MT)
Mozambique (MZ)
- ASTEPRO as AZELASTINE HYDROCHLORIDE
Netherlands (NL)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- POLLIVAL as AZELASTINE HYDROCHLORIDE
New Zealand (NZ)
Poland (PL)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- ALLESTIN as AZELASTINE HYDROCHLORIDE
- AZEL-DROP ALERGIA as AZELASTINE HYDROCHLORIDE
- AZELAMED as AZELASTINE HYDROCHLORIDE
- (combination) AZECORT as AZELASTINE HYDROCHLORIDE
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
Romania (RO)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
- (combination) SYNAZE as AZELASTINE HYDROCHLORIDE
Singapore (SG)
South Africa (ZA)
Spain (ES)
Tunisia (TN)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- AZEAL
Turkey (TR)
- ALLERGODIL as AZELASTINE HYDROCHLORIDE
- AZENOSE as AZELASTINE HYDROCHLORIDE
- NAZALASTIN as AZELASTINE HYDROCHLORIDE
- NAZETIN as AZELASTINE HYDROCHLORIDE
- ZELASS as AZELASTINE HYDROCHLORIDE
- (combination) DYMISTA as AZELASTINE HYDROCHLORIDE
United Kingdom (UK)
Note the following: The list of brand names is continuously updated, and thus does not include the total of products circulating worldwide.
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