Cabozantinib

Chemical formula: C₂₈H₂₄FN₃O₅  Molecular mass: 501.514 g/mol  PubChem compound: 25102847

Therapeutic indications

Cabozantinib is indicated for:

Renal cell carcinoma (RCC) - monotherapy

Population group: only adults (18 years old or older)

Cabozantinib is indicated as monotherapy for advanced renal cell carcinoma:

  • as first-line treatment of adult patients with intermediate or poor risk,
  • in adults following prior vascular endothelial growth factor (VEGF)-targeted therapy.

For this indication, competent medicine agencies globally authorize below treatments (click for details):

Hepatocellular carcinoma (HCC)

Population group: only adults (18 years old or older)

Cabozantinib is indicated as monotherapy for the treatment of hepatocellular carcinoma (HCC) in adults who have previously been treated with sorafenib.

For this indication, competent medicine agencies globally authorize below treatments (click for details):

Renal cell carcinoma (RCC) - combination treatment with nivolumab

Population group: only adults (18 years old or older)

Cabozantinib, in combination with nivolumab, is indicated for the first-line treatment of advanced renal cell carcinoma in adults.

For this indication, competent medicine agencies globally authorize below treatments (click for details):

Neuroendocrine tumours (NET)

Population group: only adults (18 years old or older)

Cabozantinib is indicated for the treatment of adult patients with unresectable or metastatic, well differentiated extra-pancreatic (epNET) and pancreatic (pNET) neuroendocrine tumours who have progressed following at least one prior systemic therapy other than somatostatin analogues.

For this indication, competent medicine agencies globally authorize below treatments (click for details):

Medullary thyroid carcinoma

Population group: only adults (18 years old or older)

Cabozantinib is indicated for the treatment of adult patients with progressive, unresectable locally advanced or metastatic medullary thyroid carcinoma.

For patients in whom rearranged during transfection (RET) mutation status is not known or is negative, a possible lower benefit should be taken into account before individual treatment decision.

For this indication, competent medicine agencies globally authorize below treatments (click for details):

Contraindications

Cabozantinib is contraindicated in the following cases:

Surgical procedure

Surgical procedure

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Factors such as age, gender, and health history are evaluated to create a personalized medication regimen.

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