Eletriptan

Chemical formula: C₂₂H₂₆N₂O₂S  Molecular mass: 382.519 g/mol  PubChem compound: 77993

Active ingredient description

Eletriptan is a selective agonist at the vascular 5-HT1B and neuronal 5-HT1D receptors. Eletriptan also exhibits high affinity for the 5-HT1F receptor which may contribute to its anti-migraine mechanism of action.

Medicine classification

This medicinal substance has been classified in the anatomical therapeutic chemical (ATC) classification according to its main therapeutic use as follows:

ATC code Group title Classification
N02CC06 Eletriptan N Nervous system → N02 Analgesics → N02C Antimigraine preparations → N02CC Selective serotonin (5HT1) agonists
Discover more medicines within N02CC06

Product monographs

Competent medicine agencies globally have authorized commercialization of this active ingredient according to these medication package inserts (MPIs):

Title Information Source Document Type  
RELPAX Film-coated tablet Medicines & Healthcare Products Regulatory Agency (GB) MPI, EU: SmPC

Structural formula

Graphic representation of the active ingredient's molecular structure

External identifiers

CAS Substance: 143322-58-1
DrugBank Drug: DB00216
KEGG Drug: D07887
PubChem Compound: 77993
RxNorm Ingredient: 231049
SNOMED-CT Concept: 410843003
Eletriptan (substance)
UNII Identifier: 22QOO9B8KI
ELETRIPTAN

Medicines

Eletriptan is an active ingredient of these brands:

United States (US)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Australia (AU)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Austria (AT)

  • ELETOP as ELETRIPTAN HYDROBROMIDE
  • RELPAX as ELETRIPTAN HYDROBROMIDE

Canada (CA)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Croatia (HR)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Finland (FI)

  • RELERT as ELETRIPTAN HYDROBROMIDE

France (FR)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Germany (DE)

  • ELETRIP as ELETRIPTAN HYDROBROMIDE
  • RELPAX as ELETRIPTAN HYDROBROMIDE

Hong Kong (HK)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Ireland (IE)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Israel (IL)

  • RELERT as ELETRIPTAN HYDROBROMIDE

Italy (IT)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Japan (JP)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Malta (MT)

  • ELETRIP as ELETRIPTAN HYDROBROMIDE

Mexico (MX)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Netherlands (NL)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

New Zealand (NZ)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Poland (PL)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Singapore (SG)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

South Africa (ZA)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Spain (ES)

  • RELERT as ELETRIPTAN HYDROBROMIDE
  • RELPAX as ELETRIPTAN HYDROBROMIDE

Tunisia (TN)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Turkey (TR)

  • MIGELE as ELETRIPTAN HYDROBROMIDE
  • RELPAX as ELETRIPTAN HYDROBROMIDE

United Kingdom (UK)

  • RELPAX as ELETRIPTAN HYDROBROMIDE

Note the following: The list of brand names is continuously updated, and thus does not include the total of products circulating worldwide.

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