Linzagolix

Active ingredient description

Linzagolix is a selective, non-peptide gonadotropin-releasing hormone (GnRH) receptor antagonist that inhibits endogenous GnRH signalling by binding competitively to GnRH receptors in the pituitary gland, thereby modulating the hypothalamic-pituitary-gonadal axis.

Medicine classification

This medicinal substance has been classified in the anatomical therapeutic chemical (ATC) classification according to its main therapeutic use as follows:

ATC code Group title Classification
H01CC04 H Systemic hormonal preparations, excl. Sex hormones and insulins → H01 Pituitary and hypothalamic hormones and analogues → H01C Hypothalamic hormones → H01CC Anti-gonadotropin-releasing hormones
Discover more medicines within H01CC04

Product monographs

Competent medicine agencies globally have authorized commercialization of this active ingredient according to these medication package inserts (MPIs):

Title Information Source Document Type  
YSELTY Film-coated tablet European Medicines Agency (EU) MPI, EU: SmPC

Structural formula

Graphic representation of the active ingredient's molecular structure

External identifiers

DrugBank Drug: DB17083
KEGG Drug: D11608
UNII Identifier: 7CDW97HUEX
LINZAGOLIX

Medicines

Linzagolix is an active ingredient of these brands:

Austria (AT)

  • YSELTY as Linzagolix choline

Croatia (HR)

  • YSELTY as Linzagolix choline

France (FR)

  • YSELTY as Linzagolix choline

Italy (IT)

  • YSELTY as Linzagolix choline

Lithuania (LT)

  • YSELTY as Linzagolix choline

Note the following: The list of brand names is continuously updated, and thus does not include the total of products circulating worldwide.

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