AMELUZ Gel Ref.[116233] Active ingredients: Aminolevulinic acid

Source: European Medicines Agency (EU)  Revision Year: 2026  Publisher: Biofrontera Bioscience GmbH, Hemmelrather Weg 201, 51377 Leverkusen, Germany, Tel: +49-214-87632-66, Fax: +49-214-87632-90, Email: ameluz@biofrontera.com

Product name and form

Ameluz 78 mg/g gel.

Pharmaceutical Form

Gel.

White to yellowish gel.

Qualitative and quantitative composition

One gram (g) gel contains 78 mg of 5-aminolaevulinic acid (as hydrochloride).

Excipients with known effect: One gram gel contains 2.4 mg sodium benzoate (E211), 3 mg soybean phosphatidylcholine.

For the full list of excipients, see section 6.1.

Active Ingredient

5-Aminolevulinic acid (5-ALA) is a natural biochemical precursor of heme that is metabolised in a series of enzymatic reactions to fluorescent porphyrins, particularly PPIX. 5-ALA synthesis is regulated by an intracellular pool of free heme via a negative feedback mechanism. Administration of excess exogenous 5-ALA avoids the negative feedback control, and accumulation of PPIX occurs in target tissue. In the presence of visible light, fluorescence of PPIX (photodynamic effect) in certain target tissues can be used for photodynamic diagnosis.

List of Excipients

Xanthan gum
Soybean phosphatidylcholine
Polysorbate 80
Triglycerides, medium-chain
Isopropyl alcohol
Disodium phosphate dihydrate
Sodium dihydrogen phosphate dihydrate
Sodium benzoate (E211)
Purified water

Pack sizes and marketing

One outer carton containing one aluminium tube with epoxyphenol inner lacquer and a latex seal and a screw cap of high density polyethylene. Each tube contains 2 g of gel.

Marketing authorization holder

Biofrontera Bioscience GmbH, Hemmelrather Weg 201, 51377 Leverkusen, Germany, Tel: +49-214-87632-66, Fax: +49-214-87632-90, Email: ameluz@biofrontera.com

Marketing authorization dates and numbers

EU/1/11/740/001

Date of first authorisation: 14 December 2011
Date of latest renewal: 21 November 2016

Drugs

Drug Countries
AMELUZ Austria, Estonia, Spain, France, Croatia, Ireland, Lithuania, Poland, United Kingdom, United States

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