Antazoline

Chemical formula: C₁₇H₁₉N₃  Molecular mass: 265.353 g/mol  PubChem compound: 2200

Active ingredient description

Antazoline is an antagonist of histamine H1 receptors. It selectively bind to but does not activate histamine H1 receptors, thereby blocking the actions of endogenous histamine, which subsequently leads to temporary relief of the negative symptoms brought on by histamine.

Medicine classification

This medicinal substance has been classified in the anatomical therapeutic chemical (ATC) classification according to its main therapeutic use as follows:

ATC code Group title Classification
R01AC04 Antazoline R Respiratory system → R01 Nasal preparations → R01A Decongestants and other nasal preparations for topical use → R01AC Antiallergic agents, excl. corticosteroids
Discover more medicines within R01AC04
R06AX05 Antazoline R Respiratory system → R06 Antihistamines for systemic use → R06A Antihistamines for systemic use → R06AX Other antihistamines for systemic use
Discover more medicines within R06AX05

Structural formula

Graphic representation of the active ingredient's molecular structure

External identifiers

CAS Substance: 2508-72-7
CAS Substance: 91-75-8
DrugBank Drug: DB08799
KEGG Drug: D07458
PubChem Compound: 2200
RxNorm Ingredient: 865
SNOMED-CT Concept: 373544004
Antazoline (substance)
UNII Identifier: DHA8014SS1
ANTAZOLINE

Medicines

Antazoline is an active ingredient of these brands:

Hong Kong (HK)

  • (combination) ALLERGOPOS as ANTAZOLINE PHOSPHATE
  • (combination) OPSA-HIS as ANTAZOLINE HYDROCHLORIDE

Ireland (IE)

New Zealand (NZ)

  • (combination) ALBALON-A as ANTAZOLINE PHOSPHATE

Nigeria (NG)

  • (combination) AKALLERG as ANTAZOLINE HYDROCHLORIDE
  • (combination) ALLEREX as ANTAZOLINE HYDROCHLORIDE

Poland (PL)

Romania (RO)

  • (combination) SPERSALLERG as ANTAZOLINE HYDROCHLORIDE

Singapore (SG)

  • (combination) ALOSYN as ANTAZOLINE HYDROCHLORIDE

South Africa (ZA)

  • (combination) CIBALLERGE as ANTAZOLINE HYDROCHLORIDE
  • (combination) OCULERGE as ANTAZOLINE HYDROCHLORIDE
  • (combination) SPERSALLERG as ANTAZOLINE HYDROCHLORIDE

Spain (ES)

  • (combination) ALERGOFTAL as ANTAZOLINE PHOSPHATE
  • (combination) OPTIALERG as ANTAZOLINE PHOSPHATE

Turkey (TR)

  • (combination) SULFARHIN as ANTAZOLINE HYDROCHLORIDE

United Kingdom (UK)

Note the following: The list of brand names is continuously updated, and thus does not include the total of products circulating worldwide.

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