Chemical formula: C₉H₁₇NO₂ Molecular mass: 171.237 g/mol PubChem compound: 3446
Gabapentin readily enters the brain and prevents seizures in a number of animal models of epilepsy. Gabapentin binds with high affinity to the α2δ (alpha-2-delta) subunit of voltage-gated calcium channels and it is proposed that binding to the α2δ subunit may be involved in gabapentin’s anti-seizure effects in animals.
This medicinal substance has been classified in the anatomical therapeutic chemical (ATC) classification according to its main therapeutic use as follows:
ATC code | Group title | Classification |
---|---|---|
N02BF01 | Gabapentin | N Nervous system → N02 Analgesics → N02B Other analgesics and antipyretics → N02BF Gabapentinoids |
Competent medicine agencies globally have authorized commercialization of this active ingredient according to these medication package inserts (MPIs):
Title | Information Source | Document Type | |
---|---|---|---|
NEURONTIN Capsule / Film-coated tablet / Solution | FDA, National Drug Code (US) | MPI, US: SPL/PLR | |
NEURONTIN Capsule, hard | Medicines & Healthcare Products Regulatory Agency (GB) | MPI, EU: SmPC |
Gabapentin is an active ingredient of these brands:
Albania (AL)Brazil (BR)Canada (CA)Ecuador (EC)France (FR)Israel (IL)Malta (MT)Mexico (MX)Netherlands (NL)South Africa (ZA)Spain (ES)Turkey (TR)United Kingdom (UK)Note the following: The list of brand names is continuously updated, and thus does not include the total of products circulating worldwide. |
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